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The drug is tested on Bifidobacterium ruminantium strain: fecal isolate for biotransformation. The drug concentrations were measured before and after a 12-h incubation by liquid-chromatography-coupled mass spectrometry (LC?MS)
Assay data:208 Tested
Summary
The drug is tested on Bifidobacterium longum subsp. Infantis strain: CCUG52486 for biotransformation. The drug concentrations were measured before and after a 12-h incubation by liquid-chromatography-coupled mass spectrometry (LC?MS)
Assay data:243 Tested
The drug is tested on Bifidobacterium breve strain: DSM20213 for biotransformation. The drug concentrations were measured before and after a 12-h incubation by liquid-chromatography-coupled mass spectrometry (LC?MS)
Assay data:225 Tested
The drug is tested on Bifidobacterium adolescentis strain: ATCC 15703 for biotransformation. The drug concentrations were measured before and after a 12-h incubation by liquid-chromatography-coupled mass spectrometry (LC?MS)
Assay data:247 Tested
Antitubercular activity against Mycobacterium tuberculosis H37Rv assessed as bacterial growth inhibition incubated for 7 days by microplate alamar blue assay
Assay data:2 Tested
In vivo antimycobacterial activity against Mycobacterium tuberculosis H37Rv infected in BALB/c mouse assessed as reduction in bacterial load at 300 mg/kg, po for 5 days
Assay data:1 Tested
In vivo antimycobacterial activity against Mycobacterium tuberculosis H37Rv infected in BALB/c mouse assessed as reduction in bacterial load at 200 mg/kg, po for 2 weeks
Antitubercular activity against extensively drug resistant Mycobacterium tuberculosis clinical isolates assessed as bacterial growth inhibition incubated for 6 days by resazurin based fluorescence analysis
Assay data:1 Active, 1 Activity ≤ 1 µM, 1 Tested
Antitubercular activity against multidrug resistant Mycobacterium tuberculosis clinical isolates assessed as bacterial growth inhibition incubated for 6 days by resazurin based fluorescence analysis
Antitubercular activity against Mycobacterium tuberculosis mc2 7000 assessed as bacterial growth inhibition incubated for 6 days by resazurin based fluorescence assay
Assay data:4 Active, 3 Activity ≤ 1 µM, 4 Tested
Antitubercular activity against Mycobacterium tuberculosis H37Rv expressing the luxABCDE operon infected in human THP-1 cells assessed as reduction in intracellular bacterial load incubated for 72 hrs by luminescence analysis
Assay data:1 Active, 1 Tested
Antitubercular activity against Mycobacterium tuberculosis H37Rv expressing the luxABCDE operon assessed as bacterial growth inhibition incubated for 5 days in low oxygen condition by LORA Assay
Antitubercular activity against Mycobacterium tuberculosis H37Rv expressing the luxABCDE operon assessed as bacterial growth inhibition incubated for 28 hrs in aerobic condition by luminescence analysis
Antitubercular activity against Mycobacterium tuberculosis H37Rv assessed as bacterial growth inhibition incubated for 6 days by MABA analysis
Antitubercular activity against Mycobacterium bovis BCG infected in mouse J774.A1 cells assessed as reduction in intracellular bacterial load incubated for 6 days
Assay data:1 Active, 2 Tested
Antitubercular activity against Mycobacterium tuberculosis H37Rv assessed as bacterial growth inhibition by microdilution method
Assay data:2 Active, 2 Activity ≤ 1 µM, 2 Tested
Antitubercular activity against Mycobacterium tuberculosis H37Rv assessed as bacterial growth inhibition incubated for 24 hrs by [14C]-acetate labelling based radiometric analysis
Assay data:3 Active, 3 Activity ≤ 1 µM, 3 Tested
Antitubercular activity against Mycobacterium bovis BCG assessed as bacterial growth inhibition incubated for 24 hrs by [14C]-acetate labelling based radiometric analysis
Antitubercular activity against Mycobacterium marinum strain M assessed as bacterial growth inhibition incubated for 14 days by agar plate method
Antitubercular activity against Mycobacterium bovis BCG assessed as bacterial growth inhibition incubated for 14 days by agar plate method
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